Practical synthesis of indoles and benzofurans in water using a heterogeneous bimetallic catalyst

نویسندگان

  • Cybille Rossy
  • Eric Fouquet
  • François-Xavier Felpin
چکیده

This paper describes the preparation of indoles, azaindoles and benzofurans in pure water by using a new heterogeneous Pd-Cu/C catalyst through a cascade Sonogashira alkynylation-cyclization sequence. Details of the optimization studies and the substrate scope are discussed. This procedure allows the preparation of heterocycles with good yields and is tolerant to a wide variety of functional groups.

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عنوان ژورنال:

دوره 9  شماره 

صفحات  -

تاریخ انتشار 2013